Drug name
Last update: Oct 2026Developer(s)
GS-3242 + lenacapavir
investigational
Small molecule
INSTI (Integrase Strand Transfer Inhibitor), Capsid inhibitor — INSTI+capsid inhibitor
Active / In Development (Phase 1/2/3)
Not provided
Unknown
Unknown
Oral, Subcutaneous, Route of administration is being determined in the clinical program
Aqueous drug particle suspension, Oral solid form
to be determined
to be determined
to be determined
Not provided
Not provided
Cabotegravir + Lenacapavir
lenacapavir + teropavimab + zinlirvimab
Lenacapavir 6-monthly
Lenacapavir Once-Yearly
MK-8591D (Islatravir and Lenacapavir)
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
Not provided
There are either no relevant patents or these were not yet submitted to LAPaL